137-145
| Chlorogenic Acid and Synthetic Chlorogenic Acid Derivatives: Novel Inhibitors of Hepatic Glucose-6-phosphate Translocase
Horst Hemmerle,
Hans-Joerg Burger,
Peter Below,
Gerrit Schubert,
Robert Rippel,
Peter W. Schindler,
Erich Paulus, and
Andreas W. Herling
[Full Article -
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146-167
| Structure-Activity Relationships of Selective Estrogen Receptor Modulators: Modifications to the 2-Arylbenzothiophene Core of Raloxifene
Timothy A. Grese,
Stephen Cho,
Don R. Finley,
Alexander G. Godfrey,
Charles D. Jones,
Charles W. Lugar III,
Michael J. Martin,
Ken Matsumoto,
Lewis D. Pennington,
Mark A. Winter,
M. Dee Adrian,
Harlan W. Cole,
David E. Magee,
D. Lynn Phillips,
Ellen R. Rowley,
Lorri L. Short,
Andrew L. Glasebrook, and
Henry U. Bryant
[Full Article -
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168-180
| Expeditious Syntheses of Sugar-Modified Nucleosides and Collections Thereof Exploiting Furan-, Pyrrole-, and Thiophene-Based Siloxy Dienes
Gloria Rassu,
Franca Zanardi,
Lucia Battistini,
Enrico Gaetani, and
Giovanni Casiraghi
[Full Article -
PDF] |
181-191
| Cyclic Urea Amides: HIV-1 Protease Inhibitors with Low Nanomolar Potency against both Wild Type and Protease Inhibitor Resistant Mutants of HIV
Prabhakar K. Jadhav,
Paul Ala,
Francis J. Woerner,
Chong-Hwan Chang,
Sena S. Garber,
Elizabeth D. Anton, and
Lee T. Bacheler
[Full Article -
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192-200
| Structure-Activity Relationships of Cysteine-Lacking Pentapeptide Derivatives That Inhibit ras Farnesyltransferase
Daniele M. Leonard,
Kevon R. Shuler,
Cynthia J. Poulter,
Scott R. Eaton,
Tomi K. Sawyer,
John C. Hodges,
Ti-Zhi Su,
Jeffrey D. Scholten,
Richard C. Gowan,
Judith S. Sebolt-Leopold, and
Annette M. Doherty
[Full Article -
PDF] |
201-209
| Synthesis and Inhibition Studies of Sulfur-Substituted Squalene Oxide Analogues as Mechanism-Based Inhibitors of 2,3-Oxidosqualene-Lanosterol Cyclase
Dirk Stach,
Yi Feng Zheng,
Alice L. Perez, and
Allan C. Oehlschlager
, Ikuro Abe and
Glenn D. Prestwich
, Peter G. Hartman
[Full Article -
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210-215
| Identification of High-Potency Neuropeptide Y Analogues through Systematic Lactamization
Dean A. Kirby,
Karen T. Britton,
Michel L. Aubert, and
Jean E. Rivier
[Full Article -
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216-225
| Camptothecin and Minor-Groove Binder Hybrid Molecules: Synthesis, Inhibition of Topoisomerase I, and Anticancer Cytotoxicity in Vitro
Rulin Zhao,
Naim H. Al-Said,
Daniel L. Sternbach, and
J. William Lown
[Full Article -
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226-235
| Synthesis and Protein Kinase C Inhibitory Activities of Balanol Analogs with Replacement of the Perhydroazepine Moiety
Yen-Shi Lai,
José S. Mendoza,
G. Erik Jagdmann, Jr.,
David S. Menaldino,
Christopher K. Biggers,
Julia M. Heerding,
Joseph W. Wilson,
Steven E. Hall,
Jack B. Jiang,
William P. Janzen, and
Lawrence M. Ballas
[Full Article -
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236-241
| Butitaxel Analogues: Synthesis and Structure-Activity Relationships
Syed M. Ali,
Michael Z. Hoemann,
Jeffrey Aubé,
Gunda I. Georg, and
Lester A. Mitscher
, Lalith R. Jayasinghe
[Full Article -
PDF] |
242-249
| Coumarin-Based Inhibitors of HIV Integrase
He Zhao,
Nouri Neamati,
Huixiao Hong,
Abhijit Mazumder,
Shaomeng Wang,
Sanjay Sunder,
George W. A. Milne,
Yves Pommier, and
Terrence R. Burke, Jr.
[Full Article -
PDF] |
250-259
| 3-[[(4-Aryl-1-piperazinyl)alkyl]cyclohexyl]-1H-indoles as Dopamine D2 Partial Agonists and Autoreceptor Agonists
David J. Wustrow,
William J. Smith III,
Ann E. Corbin,
M. Duff Davis,
Lynn M. Georgic,
Thomas A. Pugsley,
Steven Z. Whetzel,
Thomas G. Heffner, and
Lawrence D. Wise
[Full Article -
PDF] |
260-260
| Books of Interest
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